WIN 56,098
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| Formula | C30H28N2O2 |
| Molar mass | 448.566 g·mol−1 |
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WIN 56,098 is a chemical that is considered to be an aminoalkylindole derivative. It is a tricyclic aryl derivative that acts as a competitive antagonist at the CB2 cannabinoid receptor. Its activity at CB1 was significantly less effective. WIN 56,098 failed to antagonize any of the in vivo effects of THC.[1]
See also
References
- ^ Howlett AC, Berglund B, Melvin LS (October 1995). "Cannabinoid Receptor Agonists and Antagonists". Current Pharmaceutical Design. 1 (3): 343–352. doi:10.2174/1381612801666220918164118. S2CID 252386978.
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